《當代分子藥理學》旨在發表細胞和分子藥理學的最新進展，重點介紹正在開發的新藥物的作用機制、創新藥理學技術、細胞信號、轉導途徑分析、基因組學、蛋白質組學和代謝組學在藥物作用中的應用。另一個重點將是如何通過了解藥物在細胞和分子水平上的作用來闡明正常的生物功能。該雜志出版有關分子藥理學的專家評論、原創研究文章和專題問題。《現代分子藥理學》是一份重要的期刊，為每一位參與藥物設計和發現、目標識別、目標驗證、臨床前和臨床開發的科學家提供治療人類疾病的有用藥物。

Current Molecular Pharmacology aims to publish the latest developments in cellular and molecular pharmacology with a major emphasis on the mechanism of action of novel drugs under development, innovative pharmacological technologies, cell signaling, transduction pathway analysis, genomics, proteomics, and metabonomics applications to drug action. An additional focus will be the way in which normal biological function is illuminated by knowledge of the action of drugs at the cellular and molecular level. The journal publishes expert reviews , original research articles and thematic issues on molecular pharmacology.Current Molecular Pharmacology is an essential journal for every scientist who is involved in drug design and discovery, target identification, target validation, preclinical and clinical development of drugs therapeutically useful in human disease.